Publications

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New Antiproliferative Pyrazole/Quinoline Hybrids: Design, Synthesis, and Biological Evaluation as EGFR Inhibitors

Chemical Biology & Drug Design | 2026

DOI: https://doi.org/10.1111/cbdd.70256

Design, synthesis, in silico studies, and antiproliferative activity of a novel series of thiazole/1,2,3-triazole hybrids as apoptosis inducers and multi-kinase inhibitors endowed with anti-breast cancer activity

RSC Advances | 2026

DOI: https://doi.org/10.1039/d5ra07556d

The novel Bruton tyrosine kinase inhibitor branebrutinib abrogates lipopolysaccharide/galactosamine-induced hepatic injury via limiting inflammation and oxidative stress

Biomedicine & Pharmacotherapy | 2025

DOI: https://doi.org/10.1016/j.biopha.2025.118462

Targeting amyloid β42 aggregation using a structurally defined graphene quantum dot model: A combined molecular and biological investigation

International Journal of Biological Macromolecules | 2025

DOI: https://doi.org/10.1016/j.ijbiomac.2025.146205

New antiproliferative 1,3,4-oxadiazole/benzimidazole derivatives: Design, synthesis, and biological evaluation as dual EGFR and BRAFV600E inhibitors

Bioorganic Chemistry | 2025

DOI: https://doi.org/10.1016/j.bioorg.2025.108297

Design and synthesis of new quinoline-ester/-amide derivatives as potent antiproliferative agent targeting EGFR and BRAFV600E kinases

Journal of Molecular Structure | 2024

DOI: https://doi.org/10.1016/j.molstruc.2023.136953

Design, Synthesis and Biological Evaluation of Syn and Anti-like Double Warhead Quinolinones Bearing Dihydroxy Naphthalene Moiety as Epidermal Growth Factor Receptor Inhibitors with Potential Apoptotic Antiproliferative Action

Molecules | 2024

DOI: https://doi.org/10.3390/molecules27248765

Exploring the potential of quercetin/aspirin‑loaded chitosan nanoparticles coated with Eudragit L100 in the treatment of induced‑colorectal cancer in rats

Drug Delivery and Translational Research | 2024

DOI: https://doi.org/10.1007/s13346-023-01338-3

Novel 1,2,4-oxadiazole/pyrrolidine hybrids as DNA gyrase and topoisomerase IV inhibitors with potential antibacterial activity

Arabian Journal of Chemistry | 2024

DOI: https://doi.org/10.1016/j.arabjc.2021.103538

Optimization and SAR investigation of novel 2,3- dihydropyrazino[1,2-a] indole-1,4-dione derivatives as EGFR and BRAFV600E dual inhibitors with potent antiproliferative and antioxidant activities

Bioorganic Chemistry | 2024

DOI: https://doi.org/10.1016/j.bioorg.2022.105616

Design, synthesis, and biological evaluation of indole-2-carboxamides as SARS CoV-2 main protease inhibitors

Tetrahedron | 2023

DOI: https://doi.org/10.1016/j.tet.2023.133628

Synthesis of bis‑thiohydantoin derivatives as an antiproliferative agents targeting EGFR inhibitory pathway

Molecular Diversity | 2023

DOI: https://doi.org/10.1007/s11030-023-10653-3

Design and construction of novel pyridine-pyrimidine hybrids as selective COX-2 suppressors: anti-inflammatory potential, ulcerogenic profile, molecular modeling and ADME/Tox studies

Journal of biomolecular Structure & Dynamics | 2023

DOI: https://doi.org/10.1080/07391102.2023.2293257

Mitigation of acetaminophen-induced liver toxicity by the novel phosphatidylinositol 3-kinase inhibitor alpelisib

Front. Pharmacol | 2023

DOI: https://doi.org/10.3389/fphar.2023.1212771

Discovery of new 5-substituted-indole-2- carboxamides as dual epidermal growth factor receptor (EGFR)/cyclin dependent kinase-2 (CDK2) inhibitors with potent antiproliferative action

RSC Med. Chem | 2023

DOI: https://doi.org/10.1039/D3MD00038A

Polymeric Nanoparticles for Delivery of Natural Bioactive Agents: Recent Advances and Challenges

Polymers | 2023

DOI: https://doi.org/10.3390/polym15051123

Synthesis and Antiproliferative Potential of Thiazole and 4- Thiazolidinone Containing Motifs as Dual Inhibitors of EGFR and BRAFV600E

Molecules | 2023

DOI: https://doi.org/10.3390/molecules28247951

Design, Synthesis, and Biological Evaluation of New Indole-2-Carboxamides as Anti-Coronaviral Agents Targeting SARS CoV-2 Main Protease inhibitors

Tetrahedron | 2023

DOI: https://doi.org/10.1016/j.tet.2023.133628

Design, synthesis, docking and mechanistic studies of new thiazolyl/thiazolidinylpyrimidine-2,4-dione antiproliferative agents

Arabian Journal of Chemistry | 2023

DOI: https://doi.org/10.1016/j.arabjc.2023.104612

Emerging roles of tyrosine kinases in hepatic inflammatory diseases and therapeutic opportunities

International Immunopharmacology | 2023

DOI: https://doi.org/10.1016/j.intimp.2023.110373

Design, synthesis and antimicrobial activity of novel quinoline- 2-one hybrids as promising DNA gyrase and topoisomerase IV inhibitors

Journal of Molecular Structure | 2023

DOI: https://doi.org/10.1016/j.molstruc.2023.134902

Development of Olive Oil Containing Phytosomal Nanocomplex for Improving Skin Delivery of Quercetin: Formulation Design Optimization, In Vitro and Ex Vivo Appraisals

Pharmaceutics | 2023

DOI: https://doi.org/10.3390/pharmaceutics15041124

Design, Synthesis and Biological Evaluation of Syn and Anti-like Double Warhead Quinolinones Bearing Dihydroxy Naphthalene Moiety as Epidermal Growth Factor Receptor Inhibitors with Potential Apoptotic Antiproliferative Action

molecules | 2023

DOI: https://doi.org/ 10.3390/molecules27248765

Design, Synthesis, and Anti-Proliferative Action of Purine/Pteridine-Based Derivatives as Dual Inhibitors of EGFR and BRAFV600E

pharmaceuticals | 2023

DOI: https://doi.org/10.3390/ ph16050716

Design, synthesis, docking and mechanistic studies of new thiazolyl/thiazolidinylpyrimidine-2,4-dione antiproliferative agents

Arabian Journal of Chemistry | 2023

DOI: https://doi.org/10.1016/j.arabjc.2023.104612

Development of Olive Oil Containing Phytosomal Nanocomplex for Improving Skin Delivery of Quercetin: Formulation Design Optimization, In Vitro and Ex Vivo Appraisals

Pharmaceutics | 2023

DOI: https://doi.org/ 10.3390/pharmaceutics15041124

Discovery of new 5-substituted-indole-2- carboxamides as dual epidermal growth factor receptor (EGFR)/cyclin dependent kinase-2 (CDK2) inhibitors with potent antiproliferative action

RSC Medicinal Chemistry | 2023

DOI: https://doi.org/ 10.1039/d3md00038a

Emerging roles of tyrosine kinases in hepatic inflammatory diseases and therapeutic opportunities

International Immunopharmacology | 2023

DOI: https://doi.org/10.1016/j.intimp.2023.110373

Exploring the potential of quercetin/aspirin‑loaded chitosan nanoparticles coated with Eudragit L100 in the treatment of induced‑colorectal cancer in rats

Drug Delivery and Translational Research | 2023

DOI: https://doi.org/10.1007/s13346-023-01338-3

Polymeric Nanoparticles for Delivery of Natural Bioactive Agents: Recent Advances and Challenges

polymers | 2023

DOI: https://doi.org/10.3390/ polym15051123

Synthesis of bis‑thiohydantoin derivatives as an antiproliferative agents targeting EGFR inhibitory pathway

Molecular Diversity | 2023

DOI: https://doi.org/10.1007/s11030-023-10653-3

Design, Synthesis, and antiproliferative action of purine/pteridine-based derivatives as dual inhibitors of EGFR and BRAFV600E

Pharmaceuticals | 2023

DOI: https://doi.org/10.3390/ph16050716

Chalcone/1,3,4-Oxadiazole/Benzimidazole hybrids as novel anti-proliferative agents inducing apoptosis and inhibiting EGFR & BRAFV600E

BMC Chemistry | 2023

DOI: https://doi.org/10.1186/s13065-023-01003-3

Synthesis of novel amidines via one-pot three component reactions: Selective topoisomerase I inhibitors with antiproliferative properties

Frontiers in Chemistry | 2022

DOI: https://doi.org/10.3389/fchem.2022.1039176

New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition

Arch. Pharm. | 2022

DOI: https://doi.org/10.1002/ardp.202200024

Synthesis of novel amidines via one-pot three component reactions: Selective topoisomerase I inhibitors with antiproliferative properties

Frontiers in Chemistry | 2022

DOI: https://doi.org/10.3389/fchem.2022.1039176

Development and assessment of phospholipid-based luteolin-loaded lipid nanocapsules for skin delivery

International Journal of Pharmaceutics | 2022

DOI: https://doi.org/10.1016/j.ijpharm.2022.122375

A comprehensive review of recent advances in the biological activities of quinazolines

Chemical Biology & Drug Design | 2022

DOI: https://doi.org/10.1111/cbdd.14129

New 1,3,4‐oxadiazole‐chalcone/benzimidazole hybrids as potent antiproliferative agents

Arch. Pharm. | 2022

DOI: https://doi.org/10.1002/ardp.202200357

42- Design and synthesis of new triarylimidazole derivatives as dual inhibitors of BRAFV600E/p38α with potential antiproliferative activity

Journal of Molecular Structure | 2022

DOI: https://doi.org/10.1016/j.molstruc.2021.132218

Design, synthesis, crystal structures and biological evaluation of some 1,3-thiazolidin-4-ones as dual CDK2/EGFR potent inhibitors with potential apoptotic antiproliferative effects

Arabian Journal of Chemistry | 2022

DOI: https://doi.org/10.1016/j.arabjc.2022.104280

43- Structure-based design, synthesis and antiproliferative action of new quizoline-4-one/chalcone hybrids as EGFR inhibitors

Journal of Molecular Structure | 2022

DOI: https://doi.org/10.1016/j.molstruc.2022.132422

Development and assessment of phospholipid-based luteolin- loaded lipid nanocapsules for skin delivery

International Journal of Pharmaceutics | 2022

DOI: https://doi.org/10.1016/j.ijpharm.2022.122375

Discovery of new cyanopyridine/chalcone hybrids as dual inhibitors of EGFR/BRAFV600E with promising antiproliferative properties

Archiv der Pharmazi | 2022

DOI: https://doi.org/10.1002/ardp.202200464

New 1,3,4‐oxadiazole‐chalcone/benzimidazole hybrids as potent antiproliferative agents

Archiv der Pharmazi | 2022

DOI: https://doi.org/10.1002/ardp.202200357

46- Discovery of new pyrimido [5,4-c] quinolines as potential antiproliferative agents with multitarget actions: Rapid synthesis, docking, and ADME studies

Bioorganic Chemistry | 2022

DOI: https://doi.org/10.1016/j.bioorg.2022.105693

48- New pyrimidine/thiazole hybrids endowed with analgesic, anti-inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX/2/sEH dual inhibition

Archiv der Pharmazi | 2022

DOI: https://doi.org/10.1002/ardp.202200024

50- Novel indazole derivatives as potent apoptotic antiproliferative agents by multi-targeted mechanism: Synthesis and biological evaluation

Bioorganic Chemistry | 2022

DOI: https://doi.org/10.1016/j.bioorg.2022.105922

Design, Synthesis, and Antiproliferative Activity of Quinazolin-4-One/Chalcone Hybrids Via the Egfr Inhibition Pathway

Anti-Cancer Agents in Medicinal Chemistry | 2022

DOI: https://doi.org/10.2174/1871520623666230727104933

Mechanistic study of the antibacterial potential of the prenylated flavonoid auriculasin against Escherichia coli

Arch. Pharm. | 2022

DOI: https://doi.org/10.1002/ardp.202200360

45- New 1,3,4-oxadiazoles linked with the 1,2,3-triazole moiety as antiproliferative agents targeting the EGFR tyrosine kinase

Archiv der Pharmazi | 2022

DOI: https://doi.org/10.1002/ardp.202200009

52- Mechanistic study of the antibacterial potential of the prenylated flavonoid auriculasin against Escherichia coli

Archiv der Pharmazi | 2022

DOI: https://doi.org/10.1002/ardp.202200360

Novel indazole derivatives as potent apoptotic antiproliferative agents by multi-targeted mechanism: Synthesis and biological evaluation

Bioorganic Chemistry | 2022

DOI: https://doi.org/10.1016/j.bioorg.2022.105922

49- In Vitro Anti-Proliferative, and Kinase Inhibitory Activity of Phenanthroindolizidine Alkaloids Isolated from Tylophora indica

Plants | 2022

DOI: https://doi.org/10.3390/plants11101295

In Vitro Anti-Proliferative, and Kinase Inhibitory Activity of Phenanthroindolizidine Alkaloids Isolated fromTylophora indica

Plants | 2022

DOI: https://doi.org/10.3390/plants11101295

New 1,2,4‐oxadiazole/pyrrolidine hybrids as topoisomerase IV and DNA gyrase inhibitors with promising antibacterial activity

Arch. Pharm. | 2022

DOI: https://doi.org/10.1002/ardp.202100516

Discovery of new pyrimido[5,4-c]quinolines as potential antiproliferative agents with multitarget actions: Rapid synthesis, docking, and ADME studies

Bioorganic Chemistry | 2022

DOI: https://doi.org/10.1016/j.bioorg.2022.105693

Optimization and SAR investigation of novel 2,3-dihydropyrazino[1,2-a] indole-1,4-dione derivatives as EGFR and BRAFV600E dual inhibitors with potent antiproliferative and antioxidant activities

Bioorganic Chemistry | 2022

DOI: https://doi.org/10.1016/j.bioorg.2022.105616

Structure-based design, synthesis and antiproliferative action of new quizoline-4-one/chalcone hybrids as EGFR inhibitors

Journal of Molecular Structure | 2022

DOI: https://doi.org/10.1016/j.molstruc.2022.132422

New1,3,4?oxadiazoles linked with the 1,2,3?triazole moiety as antiproliferative agents targeting the EGFR tyrosine kinase

Arch. Pharm | 2022

DOI: https://doi.org/10.1002/ardp.202200009

Design and synthesis of new triarylimidazole derivatives as dual inhibitors of BRAF V600E /p38 ?with potential antiproliferative activity

Journal of Molecular Structure | 2021

DOI: https://doi.org/10.1016/j.molstruc.2021.132218

Design and Synthesis of (2-oxo-1,2-Dihydroquinolin-4-yl)- 1,2,3-triazole Derivatives via Click Reaction: Potential Apoptotic Antiproliferative Agents

molecules | 2021

DOI: https://doi.org/10.3390/molecules26226798

Novel 1,2,4-oxadiazole/pyrrolidine hybrids as DNA gyrase and topoisomerase IV inhibitors with potential antibacterial activity

Arabian Journal of Chemistry | 2021

DOI: https://doi.org/10.1016/j.arabjc.2021.103538

Cold-pressed raspberry seeds oil ameliorates high-fat diet triggered non-alcoholic fatty liver disease

Saudi Pharmaceutical Journal | 2021

DOI: https://doi.org/10.1016/j.jsps.2021.09.014

Discovery of novel oxazole-based macrocycles as anti-coronaviral agents targeting SARS-CoV-2 main protease

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.105363

Cold-pressed raspberry seeds oil ameliorates high-fat diet triggered non-alcoholic fatty liver disease

Saudi Pharmaceutical Journal | 2021

DOI: https://doi.org/10.1016/j.jsps.2021.09.014

Novel 1,5-diaryl pyrazole-3-carboxamides as selective COX-2/sEH inhibitors with analgesic, anti-inflammatory, and lower cardiotoxicity effects

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.105302

New quinoline/1,2,4-triazole hybrids as dual inhibitors of COX-2/5-LOX and inflammatory cytokines: Design, synthesis, and docking study

Journal of Molecular Structure | 2021

DOI: https://doi.org/10.1016/j.molstruc.2021.130948

Design, synthesis, and biological evaluation of novel EGFR inhibitors containing 5-chloro-3-hydroxymethyl-indole-2-carboxamide scaffold with apoptotic antiproliferative activity

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.104960

Design, Synthesis, and Antibacterial Screening of Some Novel Heteroaryl-Based Ciprofloxacin Derivatives as DNA Gyrase and Topoisomerase IV Inhibitors

pharmaceuticals | 2021

DOI: https://doi.org/10.3390/ph14050399

Design, synthesis, and antibacterial evaluation of new quinoline-1,3,4-oxadiazole and quinoline-1,2,4-triazole hybrids as potential inhibitors of DNA gyrase and topoisomerase IV

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.104920

Design, synthesis, and biological evaluation of new pyrimidine-5-carbonitrile derivatives bearing 1,3-thiazole moiety as novel anti-inflammatory EGFR inhibitors with cardiac safety profile

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.104890

Novel 1,2,4-triazole derivatives as apoptotic inducers targeting p53: Synthesis and antiproliferative activity

Bioorganic Chemistry | 2020

DOI: https://doi.org/10.1016/j.bioorg.2020.104369

Inhibition of Bruton tyrosine kinase by acalabrutinib dampens lipopolysaccharide/galactosamine-induced hepatic damage

Biomedicine & Pharmacotherapy | 2020

DOI: https://doi.org/10.1016/j.biopha.2020.110736

Phytoconstituents and bioactivities of the bark of Pleiogynium timorense (DC.) Leenh (Anacardiaceae)

Journal of Herbmed Pharmacology | 2020

DOI: https://doi.org/10.15171/jhp.2020.03

5-Chlorobenzofuran-2-carboxamides: From allosteric CB1 modulators to potential apoptotic antitumor agents

European Journal of Medicinal Chemistry | 2019

DOI: https://doi.org/10.1016/j.ejmech.2019.05.040

The Effect of Canertinib on Sensitivity of Cytotoxic Drugs in Tamoxifen-Resistant Breast Cancer Cells In Vitro

International Journal of Genomics | 2018

DOI: https://doi.org/10.1155/2018/7628734