Publications

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Design, synthesis, in silico studies, and antiproliferative activity of a novel series of thiazole/1,2,3-triazole hybrids as apoptosis inducers and multi-kinase inhibitors endowed with anti-breast cancer activity

RSC Advances | 2026

DOI: https://doi.org/10.1039/d5ra07556d

Design and synthesis of new quinoline-ester/-amide derivatives as potent antiproliferative agent targeting EGFR and BRAFV600E kinases

Journal of Molecular Structure | 2024

DOI: https://doi.org/10.1016/j.molstruc.2023.136953

Design, Synthesis and Biological Evaluation of Syn and Anti-like Double Warhead Quinolinones Bearing Dihydroxy Naphthalene Moiety as Epidermal Growth Factor Receptor Inhibitors with Potential Apoptotic Antiproliferative Action

Molecules | 2024

DOI: https://doi.org/10.3390/molecules27248765

Design, synthesis, and biological evaluation of indole-2-carboxamides as SARS CoV-2 main protease inhibitors

Tetrahedron | 2023

DOI: https://doi.org/10.1016/j.tet.2023.133628

Design and construction of novel pyridine-pyrimidine hybrids as selective COX-2 suppressors: anti-inflammatory potential, ulcerogenic profile, molecular modeling and ADME/Tox studies

Journal of biomolecular Structure & Dynamics | 2023

DOI: https://doi.org/10.1080/07391102.2023.2293257

Discovery of new 5-substituted-indole-2- carboxamides as dual epidermal growth factor receptor (EGFR)/cyclin dependent kinase-2 (CDK2) inhibitors with potent antiproliferative action

RSC Med. Chem | 2023

DOI: https://doi.org/10.1039/D3MD00038A

Design, Synthesis, and Biological Evaluation of New Indole-2-Carboxamides as Anti-Coronaviral Agents Targeting SARS CoV-2 Main Protease inhibitors

Tetrahedron | 2023

DOI: https://doi.org/10.1016/j.tet.2023.133628

Design, synthesis, docking and mechanistic studies of new thiazolyl/thiazolidinylpyrimidine-2,4-dione antiproliferative agents

Arabian Journal of Chemistry | 2023

DOI: https://doi.org/10.1016/j.arabjc.2023.104612

Design, synthesis and antimicrobial activity of novel quinoline- 2-one hybrids as promising DNA gyrase and topoisomerase IV inhibitors

Journal of Molecular Structure | 2023

DOI: https://doi.org/10.1016/j.molstruc.2023.134902

Development of Olive Oil Containing Phytosomal Nanocomplex for Improving Skin Delivery of Quercetin: Formulation Design Optimization, In Vitro and Ex Vivo Appraisals

Pharmaceutics | 2023

DOI: https://doi.org/10.3390/pharmaceutics15041124

Design, Synthesis and Biological Evaluation of Syn and Anti-like Double Warhead Quinolinones Bearing Dihydroxy Naphthalene Moiety as Epidermal Growth Factor Receptor Inhibitors with Potential Apoptotic Antiproliferative Action

molecules | 2023

DOI: https://doi.org/ 10.3390/molecules27248765

Design, Synthesis, and Anti-Proliferative Action of Purine/Pteridine-Based Derivatives as Dual Inhibitors of EGFR and BRAFV600E

pharmaceuticals | 2023

DOI: https://doi.org/10.3390/ ph16050716

Design, synthesis, docking and mechanistic studies of new thiazolyl/thiazolidinylpyrimidine-2,4-dione antiproliferative agents

Arabian Journal of Chemistry | 2023

DOI: https://doi.org/10.1016/j.arabjc.2023.104612

Development of Olive Oil Containing Phytosomal Nanocomplex for Improving Skin Delivery of Quercetin: Formulation Design Optimization, In Vitro and Ex Vivo Appraisals

Pharmaceutics | 2023

DOI: https://doi.org/ 10.3390/pharmaceutics15041124

Discovery of new 5-substituted-indole-2- carboxamides as dual epidermal growth factor receptor (EGFR)/cyclin dependent kinase-2 (CDK2) inhibitors with potent antiproliferative action

RSC Medicinal Chemistry | 2023

DOI: https://doi.org/ 10.1039/d3md00038a

Design, Synthesis, and antiproliferative action of purine/pteridine-based derivatives as dual inhibitors of EGFR and BRAFV600E

Pharmaceuticals | 2023

DOI: https://doi.org/10.3390/ph16050716

Development and assessment of phospholipid-based luteolin-loaded lipid nanocapsules for skin delivery

International Journal of Pharmaceutics | 2022

DOI: https://doi.org/10.1016/j.ijpharm.2022.122375

Design, synthesis, crystal structures and biological evaluation of some 1,3-thiazolidin-4-ones as dual CDK2/EGFR potent inhibitors with potential apoptotic antiproliferative effects

Arabian Journal of Chemistry | 2022

DOI: https://doi.org/10.1016/j.arabjc.2022.104280

Development and assessment of phospholipid-based luteolin- loaded lipid nanocapsules for skin delivery

International Journal of Pharmaceutics | 2022

DOI: https://doi.org/10.1016/j.ijpharm.2022.122375

Discovery of new cyanopyridine/chalcone hybrids as dual inhibitors of EGFR/BRAFV600E with promising antiproliferative properties

Archiv der Pharmazi | 2022

DOI: https://doi.org/10.1002/ardp.202200464

Design, Synthesis, and Antiproliferative Activity of Quinazolin-4-One/Chalcone Hybrids Via the Egfr Inhibition Pathway

Anti-Cancer Agents in Medicinal Chemistry | 2022

DOI: https://doi.org/10.2174/1871520623666230727104933

Discovery of new pyrimido[5,4-c]quinolines as potential antiproliferative agents with multitarget actions: Rapid synthesis, docking, and ADME studies

Bioorganic Chemistry | 2022

DOI: https://doi.org/10.1016/j.bioorg.2022.105693

Design and synthesis of new triarylimidazole derivatives as dual inhibitors of BRAF V600E /p38 ?with potential antiproliferative activity

Journal of Molecular Structure | 2021

DOI: https://doi.org/10.1016/j.molstruc.2021.132218

Design and Synthesis of (2-oxo-1,2-Dihydroquinolin-4-yl)- 1,2,3-triazole Derivatives via Click Reaction: Potential Apoptotic Antiproliferative Agents

molecules | 2021

DOI: https://doi.org/10.3390/molecules26226798

Discovery of novel oxazole-based macrocycles as anti-coronaviral agents targeting SARS-CoV-2 main protease

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.105363

Design, synthesis, and biological evaluation of novel EGFR inhibitors containing 5-chloro-3-hydroxymethyl-indole-2-carboxamide scaffold with apoptotic antiproliferative activity

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.104960

Design, Synthesis, and Antibacterial Screening of Some Novel Heteroaryl-Based Ciprofloxacin Derivatives as DNA Gyrase and Topoisomerase IV Inhibitors

pharmaceuticals | 2021

DOI: https://doi.org/10.3390/ph14050399

Design, synthesis, and antibacterial evaluation of new quinoline-1,3,4-oxadiazole and quinoline-1,2,4-triazole hybrids as potential inhibitors of DNA gyrase and topoisomerase IV

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.104920

Design, synthesis, and biological evaluation of new pyrimidine-5-carbonitrile derivatives bearing 1,3-thiazole moiety as novel anti-inflammatory EGFR inhibitors with cardiac safety profile

Bioorganic Chemistry | 2021

DOI: https://doi.org/10.1016/j.bioorg.2021.104890